It is with great enthusiasm that we write the foreword for Triazole Pharmacophore Hybrids: Synthesis and Anti-Cancer Evaluation. This comprehensive work represents a significant contribution to the fields of medicinal chemistry and oncology, focusing on the synthesis and pharmacological potential of triazole hybrids-a class of compounds with immense promise in the fight against cancer. We have observed the continuous evolution of therapeutic strategies aimed at combating cancer. Among these, triazole-based pharmacophores have garnered significant attention due to their unique chemical properties and versatile biological activities. The meticulous synthesis of these compounds and their rigorous evaluation as anti-cancer agents, as presented in this book, mark a critical step forward in advancing our understanding of their potential. The authors have masterfully synthesized a wealth of knowledge, offering insights into the design, synthesis, and biological evaluation of these hybrids. The detailed methodologies and comprehensive experimental evaluations presented herein make this book a valuable resource for both seasoned researchers and those new to the field.